Ho ruruha ka pathogen e sa tsejoeng kapa mafu a tsoakiloeng (likokoana-hloko, li-fungus), lithethefatsi tse nang le mosebetsi o moholo ka ho fetisisa o ka khonehang. 5-NOC ke setsebi sa antibacteria se rarahaneng se sebetsang khahlanong le likokoana-hloko tse tsebahalang haholo. E atleha khahlanong le li-mycoses tse ling.
5-NOC - tlhahiso
Sejo se ka sehloohong sa lithethefatsi tse potsoeng ke nitroxoline. Ke motsoako oa lik'hemik'hale o tsoang ho 8-hydroxyquinoline, o thibela ho qaptjoa ha DNA ho tloha lisele tsa likokoana-hloko 'me o thibela ho ikatisa. Lisebelisoa tse thusang tse kenyelletsoeng ho hlahisoa ha li-tablet ka 5-NOC li kenyelletsa:
- lactose monohydrate;
- calcium hydrogen phosphate;
- starch ea poone;
- Povidone K25;
- colloidal silicon dioxide;
- e hloekisitsoeng talc;
- stearate ea magnesium;
- crospovidone.
Lipilisi li hlahisoa ka khetla e sireletsang, e nang le lintho tse latelang:
- carmellose sodium;
- lemon;
- colloidal silicon dioxide;
- Povidone K25;
- titanium dioxide;
- starch ea poone;
- sucrose;
- e hloekisitsoeng talc;
- calcium carbonate;
- mebala ea lijo - mosehla "Sunset Sunset" (E110) le quinoline (E104).
5-NOC - pontšo
Moriana o reretsoe ho phekoloa ho tšoaetso e matla kapa e liehang hangata ea mekhoa ea ho ntša metsi le ea ho ikatisa. Matlapa a 5-NOC a atleha khahlanong le lihlopha tsena tsa likokoana-hloko:
- Aerobic aerobic le anaerobic;
- gram-negative aerobic le anaerobic;
- mycoplasma ;
- ureaplasma ;
- Trichomonas;
- Mycobacterium lefuba;
- dermatophyte;
- hlobo ea fungus;
- mokhethoa;
- Likokoana-hloko li baka mescoses e tebileng le e matla.
5-NOC - matšoao a sebelisoang:
- cystitis;
- pyelonephritis ;
- epididymitis;
- urethritis;
- tšoaetso e nang le tšoaetso (adenoma, carcinoma) ea prothete;
- prostatitis;
- ho ruruha ka senya kapa pampitšana e hlahang.
Ho hlophisoa ho hlalosoang ho sebelisoa ho thibela tšoaetso maemong a joalo:
- nako ea postoperative;
- ho tšoaroa ke lefu;
- cystoscopy ;
- catheterization.
5-NOC - litla-morao
Meriana e matla ea antibacteria e ka tsosa liketso tse mpe tsa 'mele ho tloha leha e le efe tsamaiso. Sena se bolela hore ka seoelo se lebisang litlamong. Liketsahalong tse ikhethang, tlhahiso ea 5-NOC e baka:
- tachycardia;
- ho hlatsa;
- anorexia;
- ho nyekeloa ke pelo;
- ho se sebetse sebete;
- botsoa;
- optic neuritis (ka tumello ea nako e telele);
- paresthesia;
- ho hloka botsitso;
- hlooho ea hlooho;
- polyneuropathy;
- thrombocytopenia;
- mefuta e mengata ea acid e ngata;
- urticaria;
- ho hlohlora letlalo;
- ataxia;
- ho senya lebese ka 'mala o mosehla o mosehla.
5-NOC ho hanyetsanoa
Sesebelisoa sena ha se khothalletsoe ho se mamellane ka bomong ho tse ling tsa lisebelisoa tse thathamisitsoeng ka holimo, ho kenyeletsoa metsoako ea lik'hemik'hale le likaroloana tsa shell. Meriana e 5-NOC e hanyetsanoa tlas'a maemo a joalo:
- ho ima;
- sebete;
- ho anyesa;
- ho ferekanngoa ho matla ha sebete kapa liphio tse nang le likhahla tse ka tlase ho 20ml / metsotsoana (e behiloeng hangata, ka hlokolosi);
- ba lilemo li ka bang 3.
U ka nka lipilisi tse 5 tsa NOC joang?
Karolo e tloaelehileng ea letsatsi le leng le le leng ea meriana e itšetlehile ka lilemo le boteng ba mafu a mang a sa foleng. Batho ba baholo ka letsatsi ba hloka 400 mg ea lithethefatsi 5-NOC - kopo e kenyeletsa ho nka tekanyo ena, e arotsoe ka makhetlo a mane, 100 mg (matlapa a mabeli) pele ho lijo. Ka lehlakoreng le matla la baktheria, karolo e habeli (800 mg). Bana ba fetang lilemo tse 5 ba fuoa meriana ea 200-400 mg ka lihora tse 24, le bana ba lilemo li 3-5 - 200 mg. Tsela e tloaelehileng ea phekolo ha ea fete libeke tse 2-4, ha ho hlokahala, e pheta hape.
Kaha ha ho na matla a ho laola le ho qhekella, 5-NOC e sebelisoa ka hlokolosi - lits'ebetso tsa tšebeliso ha li kenyelle maloetse ana, empa ka mafu a maholo, lithibela-mafu li ka etsoa. Liketsahalong tsena, nka letlapa le le leng ka makhetlo a 4 ka letsatsi. Hoa hlokahala ho hlahloba khafetsa hore na liphio le sebete li arabela joang kalafo le ho hlahloba boemo ba tumello ea creatinine.
5-NOC - kopo ea cystitis
Tekanyo ea moemeli ea antimicrobial e tšoana le tekanyo e tloaelehileng ea 400 mg nitroxoline lihora tse ling le tse ling tse 24. 5-NOC e nang le cystitis e kgothaletswa ka matsatsi a 10-21. Nako e nepahetseng ea phekolo e baloa ke urologist e thehiloeng litsing tsa laboratori, boholo ba mokhoa oa ho ruruha, le boteng ba litla-morao tsa phekolo. Ka linako tse ling e lokela ho fetisetsoa khoeli e le 'ngoe, haholo-holo haeba tšoaetso e kopantsoe kapa ea bobeli.
5-NOC e nang le pyelonephritis
Tlhaloso e hlalositsoeng ka sebōpeho se matla e hloka hore ho be le phekolo e khutšoanyane ea phekolo ea lithibela-mafu, 400 mg ka letsatsi bakeng sa libeke tse 2-2.5. Ka tsela e sa foleng ea pyelonephritis e tloaelehileng, setsebi sa urologist se etsa qeto ea ho nka 5-NOC. Ho na le merero ea phekolo ea nako e telele (likhoeli tse 2-3 bakeng sa matsatsi a 14) le mefuta e sa tšoaneng e nang le tšebeliso e telele ea lithethefatsi ka tekanyo e tlaase (100-200 mg).
Ka linako tse ling ho nka kamohelo e telele ka ho fetisisa ea 5-NOC - lipontšo bakeng sa tšebeliso e kenyeletsa mefuta e matla ea pyelonephritis:
- xanthogranulomatous;
- purulent;
- lipalo.
5-NOC nakong ea bokhachane
Ho pholletsa le nako ea bokhachane, mokhoa oa mosali oa ho ntša metsi o kotsi haholo 'me o ka hlaseloa ke ho ruruha. Ka lebaka la sena, hangata bo-'mè ba lebelloang ba thahasella 5-NOC - na nka e noa nakong ea bokhachane le litekanyetso life. Meriana-mafu ena e hanyetsanoa boemong bona, hobane e ka ama katleho kapa tlhahiso ea lesea.
5-NOC e tšoanang
Ha e hlahisa lithethefatsi tse thibelang likokoana-hloko li ke ke tsa sebelisoa kapa tsa baka litla-morao tse tebileng, e tla tlameha ho hlakoloa. Tsela feela ea ho nkela lipilisi tsa 5-NOC ke ka ho sebelisa lipoleloana tse tšoanang kapa li-generic. Ho na le litšoantšo tse peli tse tobileng ho lithethefatsi tse hlalositsoeng:
- Nitroxoline (Jeremane, Russia);
- Uroksolin (Ukraine).
Lithethefatsi tsa pele li hlahisoa ka mohopolo o fapaneng oa motsoako o sebetsang, o leng o loketseng bakeng sa phekolo e nang le litekanyetso tse phahameng. Pheko ea bobeli ke feela matlapeng a nang le lik'hemik'hale tse sebetsang tsa 50 mg. Haeba ho se lumellane le nitroxoline kapa metsoako ea eona e fumanoa, ho hlokahala hore u sebelise generic. Meriana ena e na le litšoaneleho tse tšoanang le 5-NOC - lits'ebetso tse ka sehloohong tsa tšebeliso, ts'ebetso ea antibacteria le ea boipheliso, empa sebopeho se fapaneng. Meriana e atlehang e hlahisoa ka sebōpeho sa bacteriophages:
- lefu la mali le lekaneng;
- matse;
- haeba;
- staphylococcal;
- Protheine;
- Klebsiella pneumonia;
- Pseudomonas (pseudomonas);
- kolik-proteyny;
- salmonella.
Lisebelisoa tse ling tse nang le lintlha tse tšoanang:
- Fosmicin;
- Ureacid;
- Ho tsitsa;
- Bernie;
- Fosmicin;
- Mongolo;
- Phosphoral;
- Urophosfabol;
- Boipelaetso;
- Forterase;
- Urofoscin;
- Phosphocin;
- Espa-Focine.