Timolol ke pheko ea ophthalmologic antiglaucoma, e leng lethathamong la meriana ea bohlokoa le ea bohlokoa. Nahana ka dintlha tsa motheo tsa marotholi bakeng sa mahlo a Timolol, ao mokuli ae hlokang ha a sebelisa meriana ena.
Sebopeho le mofuta oa tlhahiso ea Timolol
Ka molao, marotholi a mahlo a Timolol a fumaneha ka libotlolo tsa polasetiki-li-droppers. Karolo e sebetsang ea lithethefatsi ke timolol ka mokhoa oa maleate (maleic acid salt). Lintho tse sebetsang ka mahlaseli a mahlo a ka ba 0.5% (5 mg ea timolol ka 1 ml tharollo) kapa 0.25% (2.5 mg timolol ka 1 ml tharollo).
Li-additives bakeng sa marotholi a mahlo a timolol:
- sodium chloride;
- benzalkonium chloride;
- sodium dihydrogen phosphate dihydrate;
- disodium phosphate dodecahydrate;
- edetheate ea sodium;
- metsi a silafetseng.
Lipontšo tsa tšebeliso ea marotholi Timolol:
- ho ba le khatello ea kelello ea 'mele (khatello ea intraocular e eketsehileng);
- glaucoma e sabaletseng e sabaletseng;
- Metsoalle e koetsoeng ka mahlakoreng (e kopantsoe le maotics);
- glaucoma ea bobeli (ntle ho maikutlo, posttraumatic, aphakic);
- Congenital glaucoma (ka katleho ea mekhoa e meng ea phekolo).
Mesebetsi ea matsoho ea mahlo a marotholi a Timolol
Ntho e ka sehloohong ea lithethefatsi ke e sebetsang haholo, e sa khethollang beta-adrenergic receptor blocker (sesebelisoa se fokotsang ho ba le maikutlo a mongobo).
Phello ea lithethefatsi e bakoa haholo ke ho fokotseha ha sekhukhu sa motlakase, empa keketseho e itseng ea phallo ha e kenyelelitsoe. Litlhoko tsa timolol ha li ama boholo ba seithuti, bolulo le ho tsuba, hape li lumella ho hlahloba khatello ea "intraocular" (ophthalmotonus) nakong ea boroko.
Ho fokotsa ophthalmotonus ho finyelloa ka bobeli ka nako e tloaelehileng le ka ho eketsa khatello ea intraocular. Phello e hlokomeloa, e le molao, metsotso e 20 kamora ho sebelisoa ha lithethefatsi, e fihla holimo ka mor'a lihora tse 1 ho isa ho tse peli. Nako ea ketso ea marotholi a timolol ke hoo e ka bang lihora tse 24.
Timolol maleate e kenngoa ka potlako ka cornea. Ka tekanyo e nyenyane, lithethefatsi li kenella ho potoloha ha systemic ka ho kenngoa ka har'a lijana tsa conjunctiva le duct.
Tsela ea tsamaiso le mokhoa oa dosing timolol
Ho latela litaelo tsa tšebeliso ea marotholi a mahlo Timolol, lithethefatsi li tsamaisoa ka lerotholi le leng le le leng ka makhetlo a mabeli a metso e 'meli ka letsatsi sepakapakeng se tlaase sa leihlo le amehileng. Tlhaloso ea tharollo e khothalletsoa ke ngaka ka bomong. Haeba ho se na katleho e lekaneng, o lokela ho tsoela pele ho sebelisa tharollo e tsoetseng pele. Ka mor'a ho tsitsisa khatello ea 'mele, tekanyo ea marotholi a lithethefatsi a theoha 1 hang ka letsatsi.
Moriana o reretsoe ho sebelisoa nako e telele (ka karolelano, ho fihlela libeke tse 6). Nako ea thupelo ea phekolo e itšetlehile ka tsela ea lefu lena. Phomolo ea tšebeliso ea marotholi a timolol kapa phetoho ea tekanyo e ka phethoa feela ka khothatso ea ngaka e eang teng.
Litla-morao tsa Timolol Matotholi:
- ho fokotsa ho nyatsoa;
- corneal anesthesia;
- boemong bo botle ba ts'oaetso;
- matšoao a ho halefa habonolo.
Bakeng sa bakuli ba nang le tšebeliso ea nako e telele ea lithethefatsi, liphello tsa tsamaiso lia khoneha:
- arrhythmia;
- bradycardia;
- hypotension systemic;
- phefumoloho e khutšoanyane ;
- bronchospasm;
- botsoa.
Litlhaloso tse amanang le tšebeliso ea marotholi Timolol:
- lefu la ho fokola ha pelo;
- boloetse bo sa foleng ba pulmonary;
- sinus bradycardia;
- atrioventricular thibelo ea II le III degree;
- lefu la tsoekere;
- ho hloleha ha pelo;
- bokhachane le lactation;
- hypersensitivity ho karolo ea lithethefatsi.
Timolol - e tšoanang
Timolol ka ho buisana le ngaka e ka nkeloa sebaka ke lithethefatsi tse nang le phello e tšoanang ea meriana. Tsena li kenyelletsa:
- Khutsa;
- Fotil;
- Okumed;
- Xalatan;
- Pilocarpine;
- Betoptik.